SCHEMBL14965848

SCHEMBL14965848

CC(C)NC(=O)c1cc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cc2)ccc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.37
AVPR1B P47901 4/20 0.36
AXL P30530 2/20 0.36
MERTK Q12866 2/20 0.36
CHRM1 P11229 1/20 0.35
DHODH Q02127 1/20 0.35
KCNH2 Q12809 1/20 0.35
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
WNT1 P04628 4/20 0.34
DYRK1A Q13627 4/20 0.34
SLC2A1 P11166 1/20 0.34
EZH2 Q15910 1/20 0.34
CLK2 P49760 1/20 0.34
CLK3 P49761 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965741 0.94 MCHR1 (0.42) MCHR1AVPR1BCHRM1KCNH2NPC1
SCHEMBL14966157 0.91 AVPR1B (0.38) MCHR1AVPR1BAXLMERTK
SCHEMBL14966019 0.90 MCHR1 (0.39) MCHR1DHODHKCNH2SLC2A1
SCHEMBL14969415 0.88 HRH3 (0.42) MCHR1MEN1ALDH1A1KMT2A
SCHEMBL14965650 0.88 CNR1 (0.42) MCHR1AXLMERTKNPC1RAB9A
SCHEMBL14965822 0.88 FGFR1 (0.45) MCHR1
SCHEMBL14965639 0.88 AVPR1B (0.34) AVPR1BKCNH2
SCHEMBL14969471 0.87 KDM4E (0.41) AVPR1BSMN1; SMN2WNT1DYRK1AMEN1
SCHEMBL14965662 0.87 ALDH1A1 (0.38) MCHR1SMN1; SMN2ALDH1A1
SCHEMBL14965830 0.85 AVPR1B (0.36) MCHR1AVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed