SCHEMBL14972246

SCHEMBL14972246

COc1ccc2[nH]c(-c3ccc(-c4cnc(O[C@H]5C[C@@H](C(=O)O)C5)nc4)cc3F)nc2n1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 11/20 0.53
KCNH2 Q12809 3/20 0.46
ADORA2A P29274 2/20 0.46
PTGDR2 Q9Y5Y4 2/20 0.42
DHODH Q02127 6/20 0.40
PARP1 P09874 1/20 0.38
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14972255 0.90 DGAT1 (0.51) DGAT1KCNH2ADORA2ADHODHPARP1
SCHEMBL14972239 0.83 DGAT1 (0.47) DGAT1KCNH2ADORA2APTGDR2DHODH
SCHEMBL14972233 0.83 DGAT1 (0.45) DGAT1KCNH2ADORA2ADHODHPARP1
SCHEMBL14969110 0.81 DGAT1 (0.49) DGAT1KCNH2ADORA2ADHODH
SCHEMBL14972249 0.81 DGAT1 (0.49) DGAT1KCNH2ADORA2ADHODH
SCHEMBL14972251 0.81 DGAT1 (0.53) DGAT1KCNH2ADORA2ADHODH
SCHEMBL14971920 0.81 DHODH (0.51) DGAT1KCNH2ADORA2ADHODHPARP1
SCHEMBL14972256 0.80 DGAT1 (0.49) DGAT1KCNH2ADORA2ADHODH
SCHEMBL14971609 0.80 DGAT1 (0.47) DGAT1KCNH2ADORA2ADHODH
SCHEMBL14971563 0.80 DGAT1 (0.47) DGAT1KCNH2ADORA2ADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed