SCHEMBL14973299

SCHEMBL14973299

CCOC(=O)c1cnn(C)c1COc1ccc(F)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JMJD6 Q6NYC1 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 2/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
GAA P10253 2/20 0.40
HSP90AA1 P07900 1/20 0.40
NMT1 P30419 1/20 0.40
ALDH1A1 P00352 4/20 0.40
GPR55 Q9Y2T6 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14973111 0.85 PAX8 (0.47) JMJD6SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL14973085 0.85 ALDH1A1 (0.43) JMJD6SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL14973274 0.85 SMN1; SMN2 (0.52) SMN1; SMN2MAPTLMNAMEN1KMT2A
SCHEMBL14973126 0.83 MAPT (0.57) SMN1; SMN2MAPTLMNARAB9ANPC1
SCHEMBL14973188 0.82 TSHR (0.52) SMN1; SMN2MAPTLMNAKMT2ARAB9A
SCHEMBL14972952 0.82 MAPT (0.52) SMN1; SMN2MAPTRAB9ANPC1GAA
SCHEMBL14973272 0.82 ALDH1A1 (0.49) SMN1; SMN2MAPTLMNARAB9AGAA
SCHEMBL14973180 0.81 BRAF (0.47) SMN1; SMN2MAPTKMT2AHTTRAB9A
SCHEMBL14973032 0.81 JMJD6 (0.43) JMJD6SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL14972961 0.80 MRGPRX4 (0.43) SMN1; SMN2MAPTRAB9ANPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2604602-A1 HETEROARYL-PYRAZOLE DERIVATIVE Taisho Pharmaceutical Co., Ltd. (JP) 2013-06-19 EP disclosed
US-20130137865-A1 HETEROARYL-PYRAZOLE DERIVATIVE TAISHO PHARMACEUTICAL CO., LTD. (JP) 2013-05-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130137865-A1 HETEROARYL-PYRAZOLE DERIVATIVE GRIN2C, GRIN2B, GRIN3A JMJD6 4737/4885SMN1; SMN2 3612/4885MAPT 129/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.