SCHEMBL14975562

SCHEMBL14975562

Brc1nccn1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.49
L3MBTL1 Q9Y468 5/20 0.49
CYP1A2 P05177 5/20 0.49
CYP2D6 P10635 5/20 0.49
CYP2C9 P11712 5/20 0.49
CYP2C19 P33261 5/20 0.49
ALOX15B O15296 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.46
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
FDPS P14324 1/20 0.44
ALDH1A1 P00352 4/20 0.43
GAA P10253 1/20 0.42
CYP2E1 P05181 1/20 0.40
CYP2A6 P11509 1/20 0.40
HTT P42858 1/20 0.39
FGFR1 P11362 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28832462 0.77 NOTUM (0.51) L3MBTL1ALOX15BALDH1A1HTT
SCHEMBL25442240 0.75 NOTUM (0.46) CYP3A4L3MBTL1CYP1A2CYP2D6CYP2C9
SCHEMBL17819307 0.75 CYP19A1 (0.46)
SCHEMBL5173638 0.74 FDPS (0.47) CYP3A4L3MBTL1CYP1A2CYP2D6CYP2C9
SCHEMBL21102340 0.74 CYP3A4 (0.46) CYP3A4L3MBTL1CYP1A2CYP2D6CYP2C9
SCHEMBL2336960 0.74 CYP3A4 (0.69) CYP3A4L3MBTL1CYP1A2CYP2D6CYP2C9
SCHEMBL353826 0.74 CYP3A4 (0.50) CYP3A4L3MBTL1CYP1A2CYP2D6CYP2C9
SCHEMBL18419903 0.74 CYP3A4 (0.50) CYP3A4L3MBTL1CYP1A2CYP2D6CYP2C9
SCHEMBL10469438 0.74 CYP3A4 (0.46) CYP3A4L3MBTL1CYP1A2CYP2D6CYP2C9
SCHEMBL1407881 0.74 CYP3A4 (0.46) CYP3A4L3MBTL1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113861192-A Preparation method of C-3 halogenated imidazo [1,2-a ] pyridine derivative 郑州大学 2021-12-31 CN disclosed
CN-105793256-B Imdazole derivatives 豪夫迈·罗氏有限公司 2019-09-10 CN disclosed
CN-108473502-A 4, 6-dihydropyrrolo [3,4-C ] pyrazole-5 (1H) -carbonitrile derivatives for the treatment of cancer 特殊治疗有限公司 2018-08-31 CN disclosed
CN-105793256-A Imidazole derivatives 豪夫迈·罗氏有限公司 2016-07-20 CN disclosed
CN-104822679-A Imidazopyridine derivatives HOFFMANN LA ROCHE 2015-08-05 CN disclosed
WO-2013077654-A1 IRIDIUM (III) COMPLEX AND ORGANIC ELECTROLUMINESCENT DEVICE USING SAME 주식회사 두산 (KR) 2013-05-30 WO disclosed
CN-103097384-A Substituted imidazo [1,2-a ] pyrimidines and pyridines BAYER IP GMBH 2013-05-08 CN disclosed