SCHEMBL14975833

SCHEMBL14975833

COc1ccc(Cl)c(C#Cc2ccccc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.43
PDGFRB P09619 1/20 0.42
PDGFRA P16234 1/20 0.42
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
GRM5 P41594 7/20 0.39
KCNH2 Q12809 2/20 0.39
APP P05067 1/20 0.39
ADORA2A P29274 1/20 0.38
ADK P55263 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6821195 0.73 GRM5 (0.56) EGFRPDGFRBPDGFRAGRM5APP
SCHEMBL4858200 0.69 PDGFRB (0.46) EGFRPDGFRBPDGFRAGRM5KCNH2
SCHEMBL6133921 0.69 GRM5 (0.57) PDGFRBPDGFRAGRM5KCNH2APP
Hydrochloric Acid SCHEMBL4864461 0.68 PDGFRB (0.45) EGFRPDGFRBPDGFRAGRM5KCNH2
SCHEMBL1906166 0.67 EGFR (0.52) EGFRPDGFRBPDGFRAGRM5KCNH2
SCHEMBL15958624 0.67 GRM5 (0.48) EGFRPDGFRBPDGFRAGRM5KCNH2
SCHEMBL911440 0.67 HPGD (0.40) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL29581181 0.67 HPGD (0.40) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL1923029 0.66 ACACB (0.52) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL13865700 0.65 NNMT (0.48) PDE4APDE4BPDE4CPDE4DRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013078254-A1 BICYCLIC HETEROARYL DERIVATIVES AS KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2013-05-30 WO disclosed