SCHEMBL14979209

SCHEMBL14979209

CCc1ccc(C(=O)Nc2ccc(Cc3nn(CC(=O)O)c4ccccc34)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 8/20 0.50
TSHR P16473 1/20 0.49
ROCK1 Q13464 1/20 0.48
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
CPT1A P50416 1/20 0.46
CPT1B Q92523 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
MAPT P10636 3/20 0.45
TP53 P04637 1/20 0.45
POLB P06746 1/20 0.45
ALOX15 P16050 1/20 0.45
KDR P35968 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16153722 0.92 PTGDR2 (0.51) PTGDR2TSHRROCK1RAB9ANPC1
SCHEMBL14979185 0.90 PTGDR2 (0.51) PTGDR2TSHRROCK1CPT1ACPT1B
SCHEMBL14979170 0.86 NR1H4 (0.56) PTGDR2TSHRROCK1RAB9ANPC1
SCHEMBL14979208 0.81 L3MBTL1 (0.52) PTGDR2RAB9ANPC1HDAC3HDAC1
SCHEMBL14979173 0.78 CYP1A2 (0.51) PTGDR2RAB9ANPC1
SCHEMBL13281112 0.77 TSHR (0.61) PTGDR2TSHRALOX15
SCHEMBL16153712 0.76 NR1H4 (0.52) PTGDR2RAB9ANPC1POLB
SCHEMBL14979194 0.76 PTGDR2 (0.66) PTGDR2HDAC3HDAC1HDAC2HDAC10
SCHEMBL16085839 0.74 PTGDR2 (0.64) PTGDR2HDAC3HDAC1HDAC2HDAC10
SCHEMBL10162575 0.73 TRPV1 (0.71) RAB9ANPC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013071880-A1 NITROGEN-CONTAINING FUSED RING COMPOUNDS FOR USE AS CRTH2 ANTAGONISTS 山东亨利医药科技有限责任公司 (CN) 2013-05-23 WO disclosed