SCHEMBL14979305

SCHEMBL14979305

O=c1c(NCCCCCCOc2ccc(Cl)c(Cl)c2)c(NC2CCNCC2)c1=O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
LMNA P02545 1/20 0.38
HDAC1 Q13547 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
HRH1 P35367 2/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 2/20 0.36
UTS2R Q9UKP6 2/20 0.35
CCR3 P51677 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
ATM Q13315 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14979455 0.84 TDP1 (0.46) KDM4EALDH1A1L3MBTL1HDAC1SMN1; SMN2
SCHEMBL14979364 0.84 KDM4E (0.44) KDM4EALDH1A1L3MBTL1HDAC1GAA
SCHEMBL14979456 0.83 HDAC1 (0.41) ALDH1A1HDAC1TSHR
SCHEMBL4023510 0.74 PRKACA (0.58) KDM4EALDH1A1L3MBTL1LMNAHDAC1
SCHEMBL14979304 0.73 KDM4E (0.46) KDM4EALDH1A1L3MBTL1HDAC1SMN1; SMN2
SCHEMBL14979454 0.72 HDAC1 (0.42) KDM4EALDH1A1HDAC1SMN1; SMN2HRH1
SCHEMBL4321291 0.69 KDM4E (0.48) KDM4EALDH1A1
SCHEMBL3249653 0.68 SLC6A2 (0.63) HSP90AA1HSP90AB1
SCHEMBL19692630 0.68 ATF4 (0.59) ALDH1A1LMNASMN1; SMN2
Hydrochloric Acid SCHEMBL4156097 0.68 KDM4E (0.47) KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8450348-B2 Such as 3-[6-(4-Chloro-phenoxy)-hexylamino]-4-(pyridin-4-ylamino)-cyclobut-3-ene-1,2-dione; cancer, tumors; reduced side effects FORMA TM, LLC (US) 2013-05-28 US disclosed