SCHEMBL14979455

SCHEMBL14979455

COc1ccc(OCCCCCCNc2c(NC3CCNCC3)c(=O)c2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.46
TSHR P16473 2/20 0.46
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HDAC1 Q13547 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HPGDS O60760 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14979364 0.91 KDM4E (0.44) TSHRATML3MBTL1HDAC1KDM4E
SCHEMBL14979456 0.88 HDAC1 (0.41) TSHRHDAC1HDAC2ALDH1A1ITGB3
SCHEMBL14979305 0.84 KDM4E (0.38) TSHRATML3MBTL1HDAC1KDM4E
SCHEMBL7787085 0.80 KDM4E (0.61) TDP1KDM4EHPGDSKDM1AMAOA
SCHEMBL14979304 0.80 KDM4E (0.46) TSHRATML3MBTL1HDAC1KDM4E
SCHEMBL14979454 0.77 HDAC1 (0.42) TSHRHDAC1KDM4ESMN1; SMN2KDM1A
SCHEMBL4024280 0.72 PRKACA (0.58) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL4140224 0.68 HTR6 (0.57) TDP1TSHRL3MBTL1KDM4ESMN1; SMN2
SCHEMBL6654828 0.68 KDM4E (0.49) KDM4ESMN1; SMN2ALDH1A1CYP1A2MEN1
Hydrochloric Acid SCHEMBL27483203 0.67 GNAI3 (0.50) KDM4ESMN1; SMN2ALDH1A1CYP1A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8450348-B2 Such as 3-[6-(4-Chloro-phenoxy)-hexylamino]-4-(pyridin-4-ylamino)-cyclobut-3-ene-1,2-dione; cancer, tumors; reduced side effects FORMA TM, LLC (US) 2013-05-28 US disclosed