SCHEMBL14979872

SCHEMBL14979872

CCCCOc1c(Br)c(=O)[nH]c2c(OC)cccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
CNR2 P34972 6/20 0.46
UTS2R Q9UKP6 1/20 0.46
NQO2 P16083 1/20 0.43
KDM4E B2RXH2 4/20 0.42
MEN1 O00255 2/20 0.42
POLB P06746 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
MCL1 Q07820 2/20 0.42
LMNA P02545 1/20 0.42
BLM P54132 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HPGD P15428 3/20 0.40
ALOX12 P18054 1/20 0.40
MAPK10 P53779 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 2/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14979870 0.84 GRIN2D (0.43) CNR2SMN1; SMN2TSHR
SCHEMBL16107056 0.81 ALDH1A1 (0.50) ALDH1A1NQO2KDM4EMEN1POLB
SCHEMBL11568120 0.71 SMN1; SMN2 (0.80) ALDH1A1MEN1POLBMAPTKMT2A
SCHEMBL14979873 0.71 PARP1 (0.44) ALDH1A1CNR2KDM4EMEN1POLB
SCHEMBL12627553 0.70 SMN1; SMN2 (0.56) ALDH1A1UTS2RMEN1POLBMAPT
SCHEMBL12627551 0.69 SMN1; SMN2 (0.55) ALDH1A1UTS2RMEN1POLBMAPT
SCHEMBL14979853 0.69 MAPT (0.46) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL14376020 0.69 KDM4E (0.44) ALDH1A1CNR2UTS2RNQO2KDM4E
SCHEMBL14979958 0.68 PARP1 (0.43) ALDH1A1KDM4EHSD17B10
SCHEMBL19612454 0.68 SMN1; SMN2 (0.74) ALDH1A1MEN1POLBMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9328138-B2 HCV NS3 protease inhibitors MSD ITALIA S.R.L. (IT) 2016-05-03 US disclosed
US-20140296136-A1 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME LLC 2014-10-02 US disclosed
WO-2013074386-A2 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140296136-A1 HCV NS3 PROTEASE INHIBITORS HAVCR2, GTF3C3, CTSC ALDH1A1 1199/4885CNR2 4458/4885UTS2R 3825/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.