SCHEMBL14979870

SCHEMBL14979870

CCCCOc1c(Br)c(=O)[nH]c2c(F)cccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
GRIN1 Q05586 1/20 0.43
GRIN2A Q12879 1/20 0.43
GRIN2B Q13224 1/20 0.43
GRIN2C Q14957 1/20 0.43
GRIN3A Q8TCU5 1/20 0.43
CCNB2 O95067 2/20 0.39
CCNE2 O96020 2/20 0.39
CDK1 P06493 2/20 0.39
CDK4 P11802 2/20 0.39
CCNB1 P14635 2/20 0.39
CCND1 P24385 2/20 0.39
CCNE1 P24864 2/20 0.39
CDK2 P24941 2/20 0.39
CCND2 P30279 2/20 0.39
CCND3 P30281 2/20 0.39
CCNB3 Q8WWL7 2/20 0.39
CNR2 P34972 6/20 0.38
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14979872 0.84 ALDH1A1 (0.51) CNR2TSHRSMN1; SMN2
SCHEMBL14969170 0.80 ALDH1A1 (0.43) TSHRFEN1CTSVCTSL
SCHEMBL14979873 0.74 PARP1 (0.44) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14969214 0.70 DAO (0.49) FEN1PARP1DAODDO
SCHEMBL14979853 0.70 MAPT (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL15295256 0.70 L3MBTL1 (0.44) CCNB2CCNE2CDK1CDK4CCNB1
SCHEMBL14979851 0.70 KIF11 (0.40) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14979958 0.69 PARP1 (0.43) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14979852 0.69 MAPT (0.44) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL12596159 0.67 GRIN2D (0.38) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9328138-B2 HCV NS3 protease inhibitors MSD ITALIA S.R.L. (IT) 2016-05-03 US disclosed
US-20140296136-A1 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME LLC 2014-10-02 US disclosed
WO-2013074386-A2 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140296136-A1 HCV NS3 PROTEASE INHIBITORS HAVCR2, GTF3C3, CTSC GRIN2D 4851/4885GRIN3B 4690/4885GRIN1 4714/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.