SCHEMBL149799

SCHEMBL149799

Cc1ccc(S(=O)(=O)ONC2CN(c3ncc(OCCCC4CCN(c5ncc(Cl)cn5)CC4)cn3)CCC2c2cc(F)ccc2F)cc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 15/20 0.42
KCNH2 Q12809 7/20 0.35
CHRM2 P08172 2/20 0.34
CHRM1 P11229 2/20 0.34
CHRM3 P20309 1/20 0.34
MCHR1 Q99705 1/20 0.33
CHRM4 P08173 1/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL148875 0.87 GPR119 (0.42) GPR119KCNH2
SCHEMBL149936 0.85 GPR119 (0.34) GPR119KCNH2MCHR1SIGMAR1
SCHEMBL149798 0.85 GPR119 (0.43) GPR119KCNH2CHRM2CHRM1CHRM3
SCHEMBL120059 0.79 GPR119 (0.47) GPR119KCNH2CHRM2CHRM1CHRM3
SCHEMBL149751 0.78 GPR119 (0.42) GPR119KCNH2
SCHEMBL152138 0.78 GPR119 (0.33) GPR119KCNH2SIGMAR1
SCHEMBL149154 0.75 GPR119 (0.43) GPR119KCNH2
SCHEMBL148491 0.74 GPR119 (0.42) GPR119KCNH2
SCHEMBL150998 0.72 GPR119 (0.48) GPR119KCNH2CHRM2CHRM1CHRM3
SCHEMBL1720991 0.72 GPR119 (0.48) GPR119KCNH2CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120059014-A1 Compounds for the Treatment of Metabolic Disorders PROSIDION LIMITED (GB) 2012-03-08 US claimed
US-20120059014-A1 Compounds for the Treatment of Metabolic Disorders PROSIDION LIMITED (GB) 2012-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059014-A1 Compounds for the Treatment of Metabolic Disorders GPR119, FFAR2, GPBAR1 GPR119 1/4885KCNH2 2010/4885CHRM2 604/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.