SCHEMBL1499211

SCHEMBL1499211

N#Cc1ccc(-c2cccc([C@@H](C#N)CNC(=O)[C@@H]3CCCCN3OC(=O)C(F)(F)F)c2)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSC P53634 9/20 0.37
GPBAR1 Q8TDU6 2/20 0.35
CYP3A4 P08684 1/20 0.35
ERG P11308 1/20 0.35
CTSK P43235 3/20 0.35
CTSB P07858 2/20 0.35
CTSS P25774 2/20 0.35
SLC2A1 P11166 1/20 0.35
KCNH2 Q12809 3/20 0.35
MCHR1 Q99705 3/20 0.34
CFD P00746 1/20 0.34
BCL9 O00512 1/20 0.34
CTNNB1 P35222 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3652410 0.92 CTSC (0.42) CTSCSLC2A1MCHR1
SCHEMBL1498887 0.86 CTSC (0.37) CTSCGPBAR1CYP3A4ERGCTSK
SCHEMBL1498996 0.85 CPT2 (0.36) CTSCMCHR1
SCHEMBL3661101 0.85 MGLL (0.36) MCHR1
SCHEMBL1499150 0.85 CTSC (0.34) CTSCCTSKCTSBCTSSSLC2A1
SCHEMBL1499130 0.84 CPT2 (0.35) CTSCCTSKCTSBCTSSSLC2A1
SCHEMBL1499180 0.83 CCR3 (0.35) CTSC
SCHEMBL1499084 0.83 CTSC (0.37) CTSCCTSKCTSBCTSSBCL9
SCHEMBL3656277 0.82 DPP4 (0.38) CYP3A4MCHR1
SCHEMBL2072490 0.82 CTSC (0.49) CTSCCTSKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2011506421-A 2011-03-03 JP claimed
EP-2231597-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS AstraZeneca AB (SE) 2010-09-29 EP claimed
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO claimed