SCHEMBL1499796

SCHEMBL1499796

CC(=O)/C(=C\c1cccc([N+](=O)[O-])c1)C(=O)OC(C)C

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GLO1 Q04760 2/20 0.73
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA4 P22748 1/20 0.53
CA7 P43166 1/20 0.53
ALDH1A1 P00352 5/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
KMT2A Q03164 1/20 0.49
FBP1 P09467 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.46
MAPK1 P28482 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
HIF1A Q16665 1/20 0.44
NFE2L2 Q16236 2/20 0.43
HSP90AA1 P07900 1/20 0.43
CCR6 P51684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1499798 1.00 GLO1 (0.73) GLO1CA1CA2CA4CA7
SCHEMBL15380703 1.00 GLO1 (0.73) GLO1CA1CA2CA4CA7
SCHEMBL28927542 0.90 GLO1 (0.70) GLO1CA1CA2CA4CA7
SCHEMBL28015566 0.89 GLO1 (0.68) GLO1CA1CA2CA4CA7
SCHEMBL7275158 0.88 GLO1 (0.68) GLO1CA1CA2CA4CA7
SCHEMBL11433390 0.88 GLO1 (0.71) GLO1CA1CA2CA4CA7
SCHEMBL7275161 0.88 GLO1 (0.68) GLO1CA1CA2CA4CA7
SCHEMBL10899685 0.88 GLO1 (0.61) GLO1CA1CA2CA4CA7
SCHEMBL10665515 0.87 GLO1 (0.65) GLO1CA1CA2CA4CA7
SCHEMBL10665503 0.87 GLO1 (0.65) GLO1CA1CA2CA4CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0167068-B1 Isopropyl-2[2-(3-trifluoromethylphenoxy)ethyl]ester of 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-pyridine-3,5-dicarboxylic acid, process for its preparation, and its use as a medicine BAYER AG (DE) 1990-02-28 EP claimed
JP-11116570-A None JP disclosed
CN-106380405-A A method of synthesizing isopropyl 2-(3-nitrobenzylidene)acetoacetate 郑州瑞康制药有限公司 2017-02-08 CN disclosed
CN-106380405-A A method of synthesizing isopropyl 2-(3-nitrobenzylidene)acetoacetate 郑州瑞康制药有限公司 2017-02-08 CN disclosed
CN-102491902-A Preparation method of isopropyl 2-(3-nitrobenzylidene)acetoacetate QINGDAO HUANGHAI PHARMACEUTICAL CO LTD 2012-06-13 CN disclosed
CN-102491902-A Preparation method of isopropyl 2-(3-nitrobenzylidene)acetoacetate QINGDAO HUANGHAI PHARMACEUTICAL CO LTD 2012-06-13 CN disclosed
JP-2011201790-A MANUFACTURING METHOD OF {2-AMINO-1,4-DIHYDRO-6-METHYL-4-(3-NITROPHENYL)-3,5-PYRIDINEDICARBOXYLIC ACID 3-(1-DIPHENYLMETHYLAZETIDIN-3-YL) ESTER 5-ISOPROPYL ESTER} TOKUYAMA CORP 2011-10-13 JP disclosed
JP-2011042602-A METHOD FOR PRODUCING ISOPROPYL 2-(3-NITROBENZYLIDENE)ACETOACETATE TOKUYAMA CORP 2011-03-03 JP disclosed
JP-2011042602-A METHOD FOR PRODUCING ISOPROPYL 2-(3-NITROBENZYLIDENE)ACETOACETATE TOKUYAMA CORP 2011-03-03 JP disclosed
US-7795281-B2 Optically active dihydropyridine derivative DAIICHI SANKYO COMPANY, LIMITED (JP) 2010-09-14 US disclosed
US-3971790-A VASODILATION, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DT) 1976-07-27 US disclosed
US-3971791-A VASODILATION, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DT) 1976-07-27 US disclosed
US-3959292-A HYPOTENSIVE AGENTS, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US disclosed
US-3951994-A HYPOTENSIVE, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-04-20 US disclosed
US-3951988-A HYPOTENSIVE, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-04-20 US disclosed
US-3948923-A HYPOTENSIVE, VASODILATION BAYER AKTIENGESELLSCHAFT (DT) 1976-04-06 US disclosed
US-3946026-A HYPOTENSIVE AGENTS, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-03-23 US disclosed
US-3939171-A HYPOTENSIVE, VASODILATION BAYER AKTIENGESELLSCHAFT (DT) 1976-02-17 US disclosed
US-3935220-A VASODILATION, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DT) 1976-01-27 US disclosed
US-3935223-A 2-Amino-1,4-dihydropyridine derivatives BAYER AKTIENGESELLSCHAFT (DT) 1976-01-27 US disclosed