SCHEMBL15020409

SCHEMBL15020409

CC1c2cccnc2CCN1C=O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.39
CYP19A1 P11511 3/20 0.36
CYP2D6 P10635 1/20 0.36
TRPC3 Q13507 1/20 0.36
TRPC6 Q9Y210 1/20 0.36
TBXAS1 P24557 3/20 0.34
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
OPRK1 P41145 2/20 0.33
TMEM97 Q5BJF2 2/20 0.33
SIGMAR1 Q99720 2/20 0.33
LHCGR P22888 2/20 0.33
TRPM8 Q7Z2W7 2/20 0.33
CYP2C8 P10632 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL34469114 0.78 PPARG (0.37) PPARGCYP19A1CYP2D6TBXAS1HTR2A
SCHEMBL31569261 0.78 HRH1 (0.37) PPARGCYP19A1CYP2D6TBXAS1HTR2A
SCHEMBL15222063 0.78 MAOA (0.40) CYP19A1CYP2D6TRPC3TRPC6TBXAS1
SCHEMBL8034390 0.78 MAOA (0.40) CYP19A1CYP2D6TRPC3TRPC6TBXAS1
SCHEMBL15019739 0.76 TRPM8 (0.35) PPARGTRPM8
SCHEMBL29785644 0.74 DRD1 (0.45) HTR2AHTR2CHTR2BSIGMAR1TRPM8
SCHEMBL29676795 0.74 DRD1 (0.45) HTR2AHTR2CHTR2BSIGMAR1TRPM8
SCHEMBL20358479 0.74 DRD1 (0.45) HTR2AHTR2CHTR2BSIGMAR1TRPM8
SCHEMBL31569049 0.74 TRPC3 (0.45) TRPC3TRPC6TBXAS1HTR2AHTR2C
SCHEMBL31569530 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013087808-A1 PHARMACEUTICAL COMPOSITION COMPRISING A PYRAZOLOPYRIMIDME AND CYCLODEXTRIN MERZ PHARMA GMBH & CO. KGAA (DE) 2013-06-20 WO disclosed