SCHEMBL15028217

SCHEMBL15028217

COc1cccc(CNC(=O)c2cccc(OC3CCNCC3)c2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 3/20 0.67
CHRM3 P20309 1/20 0.62
LMNA P02545 1/20 0.60
HPGD P15428 1/20 0.60
EPHX2 P34913 1/20 0.58
MEN1 O00255 1/20 0.56
USP2 O75604 1/20 0.56
ALDH1A1 P00352 1/20 0.56
GAA P10253 1/20 0.56
KMT2A Q03164 1/20 0.56
ROCK2 O75116 4/20 0.56
AURKA O14965 1/20 0.55
MAPK14 Q16539 1/20 0.52
ROCK1 Q13464 3/20 0.52
PRKACA P17612 2/20 0.52
PRKX P51817 2/20 0.52
PRKCQ Q04759 2/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9416645 0.84 MMP13 (0.94) MMP13LMNAHPGDMEN1USP2
SCHEMBL4664685 0.83 MAPK14 (0.60) MMP13CHRM3LMNAHPGDROCK2
SCHEMBL15012854 0.82 NMT1 (0.65) MEN1KMT2AHRH1
SCHEMBL31061610 0.81 MMP13 (1.00) MMP13LMNAHPGDMEN1USP2
SCHEMBL5332068 0.81 MMP13 (1.00) MMP13LMNAHPGDMEN1USP2
SCHEMBL15028387 0.80 NMT1 (0.80) USP2
SCHEMBL13746152 0.79 ALDH1A1 (0.74) MMP13LMNAEPHX2ALDH1A1KMT2A
SCHEMBL30475500 0.78 HPGD (0.61) MMP13CHRM3LMNAHPGDALDH1A1
SCHEMBL12813045 0.78 MMP13 (0.82) MMP13LMNAHPGDMEN1USP2
SCHEMBL2807802 0.78 EPHX2 (0.55) EPHX2GSK3BHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013083991-A1 NOVEL COMPOUNDS AND THEIR USE IN THERAPY IMPERIAL INNOVATIONS LIMITED (GB) 2013-06-13 WO disclosed