SCHEMBL1503171

SCHEMBL1503171

Cc1c(C(=O)O)cnc(C(=O)O)c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.43
GABRD O14764 2/20 0.43
GABRA1 P14867 2/20 0.43
GABRB1 P18505 2/20 0.43
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
GABRA5 P31644 2/20 0.43
GABRA3 P34903 2/20 0.43
GABRA2 P47869 2/20 0.43
GABRB2 P47870 2/20 0.43
GABRA4 P48169 2/20 0.43
GABRE P78334 2/20 0.43
GABRA6 Q16445 2/20 0.43
GABRG1 Q8N1C3 2/20 0.43
GABRG3 Q99928 2/20 0.43
GABRQ Q9UN88 2/20 0.43
KDM4E B2RXH2 7/20 0.42
KMT2A Q03164 1/20 0.42
HPGD P15428 2/20 0.41
LDHA P00338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12444329 0.84 NPSR1 (0.39) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL600482 0.83 GABRP (0.46) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL28241145 0.78 KDM4E (0.47) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22283906 0.74 KDM4E (0.37) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7666078 0.73 LDHA (0.36) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL24257694 0.71 FYN (0.40)
SCHEMBL30546823 0.71 FYN (0.40)
SCHEMBL9787552 0.70 SELL (0.38) KDM4EKMT2AHPGDALDH1A1L3MBTL1
SCHEMBL31032542 0.70 SELL (0.38) KDM4EKMT2AHPGDALDH1A1L3MBTL1
SCHEMBL13313461 0.69 HPGD (0.46) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP disclosed
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO disclosed