SCHEMBL1503260

SCHEMBL1503260

O=C(NO)c1ncc(CN(c2ccc(F)cc2)C2CC2)c(CO)c1O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 10/20 0.36
HDAC3 O15379 7/20 0.36
HDAC8 Q9BY41 6/20 0.36
HRH3 Q9Y5N1 1/20 0.32
HDAC1 Q13547 5/20 0.31
HDAC2 Q92769 5/20 0.31
HDAC11 Q96DB2 3/20 0.31
HDAC4 P56524 2/20 0.31
HDAC7 Q8WUI4 2/20 0.31
HDAC10 Q969S8 2/20 0.31
HDAC9 Q9UKV0 2/20 0.31
HDAC5 Q9UQL6 2/20 0.31
TRPA1 O75762 1/20 0.31
EGLN2 Q96KS0 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31
MAOA P21397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1503183 0.79 NAMPT (0.39)
SCHEMBL2216328 0.78 EGFR (0.41) HDAC6HDAC3HDAC8HDAC1HDAC11
SCHEMBL2146957 0.77 HDAC6 (0.37) HDAC6HDAC3HDAC8HDAC1HDAC2
SCHEMBL30954811 0.76 MMP1 (0.39) EGLN1
SCHEMBL1503250 0.76 MMP1 (0.39) EGLN1
SCHEMBL1503241 0.76 HDAC1 (0.39) HDAC6HDAC3HDAC8HDAC1HDAC2
SCHEMBL1503199 0.76 ALDH1A1 (0.35) HDAC6HDAC3HDAC8HDAC1HDAC2
SCHEMBL1503231 0.75 ALDH1A1 (0.42) HDAC6HDAC3HDAC1HDAC2EGLN2
SCHEMBL1503246 0.75 EGFR (0.36) HDAC6HDAC3HDAC8HDAC1HDAC2
SCHEMBL12516709 0.74 HDAC1 (0.43) HDAC6HDAC3HDAC8HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP disclosed
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO disclosed