SCHEMBL15037702

SCHEMBL15037702

ICc1ccc(-c2ccncc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.55
LMNA P02545 1/20 0.55
CYP17A1 P05093 10/20 0.48
CYP11B1 P15538 9/20 0.48
CYP11B2 P19099 8/20 0.48
CYP3A4 P08684 6/20 0.48
CYP19A1 P11511 5/20 0.48
NOTUM Q6P988 1/20 0.46
CYP21A2 P08686 1/20 0.46
LSS P48449 1/20 0.46
KIF11 P52732 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
QDPR P09417 1/20 0.41
PRKCI P41743 1/20 0.41
CYP2D6 P10635 1/20 0.41
MMP12 P39900 1/20 0.41
MMP13 P45452 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3628639 0.84
SCHEMBL679947 0.84 HRH3 (0.47) LMNACYP17A1CYP11B1CYP11B2CYP3A4
Hydrochloric Acid SCHEMBL17654197 0.81
SCHEMBL5226620 0.80 MAPT (0.55) MAPTLMNACYP17A1CYP11B1CYP11B2
SCHEMBL10000032 0.78 MAPT (0.92) MAPTLMNACYP3A4NOTUMKIF11
SCHEMBL135626 0.78 MAPT (0.92) MAPTLMNACYP3A4NOTUMKIF11
SCHEMBL19567238 0.76 CYP2A6 (0.67) MAPTLMNACYP17A1CYP11B1CYP11B2
SCHEMBL1129630 0.75 MAPT (0.55) MAPTLMNACYP17A1CYP11B1CYP11B2
SCHEMBL8239917 0.75 MAPT (0.59) MAPTLMNACYP17A1CYP11B1CYP11B2
SCHEMBL1439245 0.75 MKNK1 (0.61) MAPTLMNACYP17A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2604269-A1 1,4-benzodiazepine-2,5-diones with therapeutic properties THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-06-19 EP disclosed