SCHEMBL1504639

SCHEMBL1504639

CC(NCC(=O)OC(C)(C)C)C(C(=O)O)N1CCN(S(C)(=O)=O)CC1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
POLB P06746 2/20 0.31
MAPK1 P28482 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ADAM17 P78536 1/20 0.31
TP53 P04637 1/20 0.31
ALDH1A1 P00352 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1504675 0.81 PREP (0.37) MEN1KMT2APOLBMAPK1CASP1
SCHEMBL10276757 0.78 ADAM17 (0.38) ADAM17
SCHEMBL995255 0.69 ADAM17 (0.43) MEN1KMT2AADAM17
SCHEMBL995012 0.69 ADAM17 (0.43) MEN1KMT2AADAM17
SCHEMBL995014 0.69 ADAM17 (0.43) MEN1KMT2AADAM17
SCHEMBL12077753 0.69 TP53 (0.33) MEN1KMT2APOLBADAM17TP53
SCHEMBL1504588 0.69 ALDH1A1 (0.41) MEN1KMT2APOLBMAPK1CASP1
SCHEMBL24269352 0.68 CYP2D6 (0.44) TDP1
Hydrochloric Acid SCHEMBL1504593 0.68 ALDH1A1 (0.40) MEN1KMT2APOLBMAPK1CASP1
Hydrochloric Acid SCHEMBL1504752 0.68 ALDH1A1 (0.40) MEN1KMT2APOLBMAPK1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011033009-A1 N- [2-HYDROXYCARBAMOYL-2- (PIPERAZINYL) ETHYL] BENZAMIDE COMPOUNDS, THEIR PREPARATION AND THEIR USE AS TACE INHIBITORS GALDERMA RESEARCH & DEVELOPMENT (FR) 2011-03-24 WO disclosed