SCHEMBL15046450

SCHEMBL15046450

Cc1cc(-c2cn(-c3ccccc3)c(CC(N)=O)n2)ccc1F

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
SRC P12931 2/20 0.47
GRM5 P41594 11/20 0.43
MAPT P10636 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.39
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA5A P35218 1/20 0.38
CA5B Q9Y2D0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15046474 0.91 ALDH1A1 (0.45) ALDH1A1SRCGRM5MAPTCA1
SCHEMBL15034007 0.91 ALDH1A1 (0.49) ALDH1A1SRCGRM5MAPTNPC1
SCHEMBL15034000 0.86 ALDH1A1 (0.48) ALDH1A1SRCGRM5MAPTNPC1
SCHEMBL15033935 0.83 GRM5 (0.43) ALDH1A1SRCGRM5MAPTCA1
SCHEMBL15046477 0.81 GRM5 (0.43) ALDH1A1SRCGRM5MAPTCA1
SCHEMBL15034561 0.79 GRM5 (0.67) GRM5KDM4ELMNA
SCHEMBL15046451 0.78 MEN1 (0.53) ALDH1A1MAPTNPC1RAB9AKDM4E
SCHEMBL15034558 0.78 GRM5 (0.68) ALDH1A1GRM5KDM4EMEN1KMT2A
SCHEMBL15034565 0.78 GRM5 (0.68) GRM5
SCHEMBL15033972 0.78 GRM5 (0.62) ALDH1A1SRCGRM5MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013087806-A1 PIPERAZINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLU5 RECEPTORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-20 WO disclosed