SCHEMBL15046477

SCHEMBL15046477

CC(=O)Cc1nc(-c2ccc(F)c(C)c2)cn1-c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.43
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
SRC P12931 2/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CA2 P00918 2/20 0.39
CA1 P00915 1/20 0.39
CA5A P35218 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
ABCB1 P08183 1/20 0.38
MAPT P10636 2/20 0.37
GRIN2B Q13224 3/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15033935 0.91 GRM5 (0.43) GRM5GABRA2GABRB2SRCPTGS1
SCHEMBL15046474 0.90 ALDH1A1 (0.45) GRM5GABRA2GABRB2SRCPTGS1
SCHEMBL15043866 0.88 GABRB2 (0.45) GABRA2GABRB2PTGS1ALDH1A1ABCB1
SCHEMBL15033983 0.87 GABRA2 (0.48) GRM5GABRA2GABRB2SRCPTGS1
SCHEMBL15046472 0.86 ABCB1 (0.49) GABRA2GABRB2PTGS1ALDH1A1ABCB1
SCHEMBL15034007 0.83 ALDH1A1 (0.49) GRM5SRCPTGS1PTGS2ALDH1A1
SCHEMBL15046450 0.81 ALDH1A1 (0.55) GRM5SRCALDH1A1CA2CA1
SCHEMBL15046476 0.81 MAPT (0.52) GABRA2GABRB2ALDH1A1MAPT
SCHEMBL15033933 0.80 PTGS1 (0.41) GRM5GABRA2GABRB2PTGS1PTGS2
SCHEMBL15034542 0.79 GRM5 (0.61) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013087806-A1 PIPERAZINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLU5 RECEPTORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-20 WO disclosed