SCHEMBL15048857

SCHEMBL15048857

Cc1ccc(-c2cccc(C(=O)O)c2-n2nncc2C(C)C)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
GAA P10253 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
BRS3 P32247 6/20 0.40
MCL1 Q07820 1/20 0.35
BAD Q92934 1/20 0.35
HSD11B1 P28845 1/20 0.35
HNF4A P41235 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 1/20 0.34
MYC P01106 1/20 0.34
AKR1C3 P42330 1/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14931575 0.72 PPARG (0.45)
SCHEMBL2276901 0.70 P2RY14 (0.42) GAAHSD11B1KDM4EALDH1A1
SCHEMBL3659233 0.69 NPC1 (0.41) NPC1GAARAB9AKMT2ABRS3
SCHEMBL372 0.68 KMT2A (0.60) NPC1GAARAB9AKMT2ABRS3
SCHEMBL31402608 0.68 KMT2A (0.60) NPC1GAARAB9AKMT2ABRS3
SCHEMBL11142513 0.67 POLB (0.54) NPC1GAARAB9AKMT2ABRS3
Hydrochloric Acid SCHEMBL7610390 0.67 KMT2A (0.59) NPC1GAARAB9AKMT2ABRS3
SCHEMBL1854636 0.67 NPC1 (0.46) NPC1GAARAB9AKMT2ABRS3
SCHEMBL15664279 0.66 POLB (0.49) NPC1GAARAB9AKMT2ABRS3
SCHEMBL17965677 0.66 TSHR (0.52) NPC1GAARAB9AKMT2ABRS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2607356-A1 Triazole-substituted arylamide derivatives and their use as P2x3 and /or P2x2/3 purinergic receptor antagonists F. Hoffmann-La Roche AG (CH) 2013-06-26 EP disclosed