SCHEMBL15054545

SCHEMBL15054545

COC(=O)C1(c2cccc([N+](=O)[O-])c2)CCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
NPSR1 Q6W5P4 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2C9 P11712 1/20 0.46
KDM1A O60341 1/20 0.45
ADRA1D P25100 4/20 0.44
ADRA1A P35348 4/20 0.44
ADRA1B P35368 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
LMNA P02545 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CHRNA1 P02708 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15054977 0.97 MEN1 (0.48) SLC6A4MEN1KMT2ANPSR1CYP1A2
SCHEMBL15054845 0.94 KDM1A (0.47) SLC6A4MEN1KMT2ANPSR1KDM1A
SCHEMBL6676255 0.83 AKR1C1 (0.53) MEN1KMT2ANPSR1CYP1A2CYP2C19
SCHEMBL3227451 0.83 MEN1 (0.58) MEN1KMT2ANPSR1CYP1A2CYP2C19
SCHEMBL8097387 0.82 ALDH1A1 (0.50) MEN1KMT2ANPSR1CYP1A2CYP2C19
SCHEMBL6676866 0.80 AKR1C1 (0.57) MEN1KMT2ANPSR1CYP1A2CYP2C19
SCHEMBL27256555 0.79 NPSR1 (0.46) SLC6A4MEN1KMT2ANPSR1CYP1A2
SCHEMBL6674979 0.79 AKR1C1 (0.56) MEN1KMT2ANPSR1CYP1A2CYP2C19
SCHEMBL2847573 0.79 HDAC4 (0.46) SLC6A4SLC6A2
SCHEMBL30492221 0.78 KDM1A (0.50) MEN1KMT2ANPSR1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096151-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2013-06-27 WO disclosed