SCHEMBL15055488

SCHEMBL15055488

O=Cc1ccc(Oc2ccc(Cl)cc2)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.47
TTR P02766 2/20 0.47
ALDH1A1 P00352 6/20 0.46
HPGD P15428 3/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TACR2 P21452 1/20 0.43
PNLIP P16233 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
EPAS1 Q99814 4/20 0.40
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30628472 0.85 TTR (0.57) HSD17B10TTRALDH1A1HPGDMAPT
SCHEMBL21190855 0.84 ALDH1A1 (0.49) TTRALDH1A1HPGDMEN1KMT2A
SCHEMBL24512660 0.83 TTR (0.60) HSD17B10TTRALDH1A1HPGDMAPT
SCHEMBL203768 0.83 TTR (0.64) TTRALDH1A1MAPTMEN1KMT2A
SCHEMBL25047358 0.81 ALDH1A1 (0.49) HSD17B10TTRALDH1A1HPGDMAPT
SCHEMBL23120903 0.81 HSD17B10 (0.47) HSD17B10TTRALDH1A1HPGDMAPT
SCHEMBL18304466 0.80 MAPT (0.49) TTRALDH1A1HPGDMAPTMEN1
SCHEMBL16791716 0.80 TTR (0.50) HSD17B10TTRALDH1A1HPGDMAPT
SCHEMBL2991888 0.80 GAA (0.53) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL26936729 0.79 TTR (0.72) TTRALDH1A1HPGDMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed
WO-2013093688-A1 SULFONAMIDE DERIVATIVES AND USE THEREOF AS VGSC INHIBITORS PFIZER LIMITED (GB) 2013-06-27 WO disclosed
WO-2013093688-A1 SULFONAMIDE DERIVATIVES AND USE THEREOF AS VGSC INHIBITORS PFIZER LIMITED (GB) 2013-06-27 WO disclosed