SCHEMBL15057413

SCHEMBL15057413

COC(=O)CC1CCC(c2ccc(-c3ccc(-c4nc(-c5ccccc5)c[nH]4)cn3)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.60
ADORA2A P29274 3/20 0.43
KCNH2 Q12809 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15057412 1.00 DGAT1 (0.60) DGAT1ADORA2AKCNH2
SCHEMBL16787660 0.89 DGAT1 (0.52) DGAT1ADORA2AKCNH2
SCHEMBL15058508 0.89 DGAT1 (0.61) DGAT1ADORA2AKCNH2
SCHEMBL15058509 0.89 DGAT1 (0.61) DGAT1ADORA2AKCNH2
SCHEMBL16790068 0.85 DGAT1 (0.57) DGAT1ADORA2AKCNH2
SCHEMBL10188659 0.80 DGAT1 (0.56) DGAT1
SCHEMBL898526 0.79 DGAT1 (0.54) DGAT1
SCHEMBL15054761 0.79 DGAT1 (0.54) DGAT1
SCHEMBL180599 0.79 DGAT1 (0.54) DGAT1
SCHEMBL180547 0.79 DGAT1 (0.54) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096093-A1 COMPOUNDS AS DGAT-1 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-06-27 WO disclosed