SCHEMBL1505819

SCHEMBL1505819

Cc1ccc(COS(C)(=O)=O)c(=O)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 9/20 0.33
HSD17B10 Q99714 5/20 0.33
HPGD P15428 3/20 0.33
HMBS P08397 1/20 0.33
MAPT P10636 3/20 0.33
KMT2A Q03164 3/20 0.32
L3MBTL1 Q9Y468 3/20 0.32
MEN1 O00255 2/20 0.32
PKM P14618 1/20 0.32
CYP1A2 P05177 2/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
SPR P35270 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1738125 0.73 HMBS (0.46) ALDH1A1KDM4EHSD17B10HPGDHMBS
Hydrochloric Acid SCHEMBL5709777 0.71 HMBS (0.43) ALDH1A1KDM4EHSD17B10HPGDHMBS
SCHEMBL20160825 0.70 HMBS (0.42) MAPK1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL2904372 0.70 GRIA1 (0.43) ALDH1A1KDM4EHSD17B10HPGDHMBS
SCHEMBL5273095 0.69 CYP1A2 (0.41) ALDH1A1KDM4EHPGDKMT2AMEN1
Hydrochloric Acid SCHEMBL5010692 0.68 HMBS (0.40) MAPK1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL20565249 0.68 EGFR (0.35) HPGDKMT2AL3MBTL1CYP1A2CYP3A4
SCHEMBL19974316 0.67 MAOB (0.44) ALDH1A1KMT2AMEN1CYP1A2CYP3A4
SCHEMBL22904635 0.66 HMBS (0.37) ALDH1A1KDM4EHSD17B10HPGDHMBS
SCHEMBL6301740 0.66 KDM4A (0.38) ALDH1A1HPGDMAPTKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2475676-A2 Pregnane derivatives condensed in the 16,17 position with an N-substituted isoxazolidine ring as anti-inflammatory agents Chiesi Farmaceutici S.p.A. (IT) 2012-07-18 EP disclosed
WO-2011029547-A2 PREGNANE DERIVATIVES CONDENSED IN THE 16, 17 POSITION WITH AN N-SUBSTITUTED ISOXAZOLIDINE RING AS ANTI-INFLAMMATORY AGENTS CHIESI FARMACEUTICI S.P.A. (IT) 2011-03-17 WO disclosed