SCHEMBL20160825

SCHEMBL20160825

Cc1ccc(CN)c(=O)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMBS P08397 1/20 0.42
SPR P35270 1/20 0.36
PARP1 P09874 1/20 0.35
KDM4E B2RXH2 5/20 0.34
GAA P10253 1/20 0.34
PKM P14618 1/20 0.34
MAPK1 P28482 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.32
DAO P14920 2/20 0.32
ALDH1A1 P00352 4/20 0.32
HSD17B10 Q99714 3/20 0.32
HPGD P15428 2/20 0.32
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5010692 0.98 HMBS (0.40) HMBSSPRPARP1KDM4EGAA
SCHEMBL1738125 0.82 HMBS (0.46) HMBSSPRKDM4EGAAPKM
Hydrochloric Acid SCHEMBL5709777 0.80 HMBS (0.43) HMBSSPRKDM4EGAAPKM
SCHEMBL2904372 0.78 GRIA1 (0.43) HMBSSPRPARP1KDM4EGAA
SCHEMBL22904635 0.74 HMBS (0.37) HMBSSPRKDM4EGAAPKM
SCHEMBL16344799 0.72 KDM4E (0.41) PARP1KDM4EGAAPKMMAPK1
SCHEMBL2690132 0.72 ALDH1A1 (0.38) PARP1KDM4EGAALOXL2DAO
SCHEMBL17238980 0.70
SCHEMBL21564300 0.70 DAO (0.37) HMBSSPRKDM4EGAAMEN1
SCHEMBL1505819 0.70 MAPK1 (0.36) HMBSSPRKDM4EPKMMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154314-A1 SPIRO PIPERIDINE DERIVATIVES AS INHIBITORS OF APOL1 AND METHODS OF USING SAME VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-08-17 WO disclosed
WO-2018086589-A1 1,5,7-TRI-SUBSTITUTED ISOQUINOLINE DERIVATIVES, PREPARATION THEREOF, AND USE THEREOF IN MEDICINES 上海海雁医药科技有限公司 2018-05-17 WO disclosed