SCHEMBL15062012

SCHEMBL15062012

Cc1ccc(F)cc1O[C@H]1CCN(C(C)C)C1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.45
SLC6A4 P31645 1/20 0.43
SCD O00767 2/20 0.40
HRH1 P35367 1/20 0.40
CCR3 P51677 1/20 0.40
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
OXTR P30559 2/20 0.39
AVPR1A P37288 2/20 0.39
AVPR2 P30518 1/20 0.39
PDE9A O76083 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
ACACB O00763 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062019 1.00 HRH3 (0.45) HRH3SLC6A4SCDHRH1CCR3
SCHEMBL15062011 0.92 HRH3 (0.46) HRH3SCDHRH1CCR3
SCHEMBL1927682 0.85 SCD (0.47) HRH3SLC6A4SCD
SCHEMBL17955442 0.83 SLC6A4 (0.43) HRH3SLC6A4SCDHTR2CHTR2B
SCHEMBL17955447 0.83 SLC6A4 (0.43) HRH3SLC6A4SCDHTR2CHTR2B
SCHEMBL15062023 0.83 HTR2C (0.54) SLC6A4SCDHTR2CHTR2BOXTR
SCHEMBL22545206 0.83 HRH3 (0.48) HRH3SCDOXTRAVPR1APDE9A
SCHEMBL15062015 0.83 HTR2C (0.54) SLC6A4SCDHTR2CHTR2BOXTR
SCHEMBL1928720 0.83 SLC6A4 (0.43) HRH3SLC6A4SCDHRH1CCR3
SCHEMBL15061995 0.81 SCD (0.47) HRH3SCDHTR2CHTR2BOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013091773-A1 TETRAAZA-CYCLOPENTA[A]INDENYL AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS MERCK PATENT GMBH (DE) 2013-06-27 WO disclosed
EP-2607364-A1 Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators Ares Trading S.A. (CH) 2013-06-26 EP disclosed