SCHEMBL15067255

SCHEMBL15067255

NS(=O)(=O)c1cnc(Oc2ccc(F)cc2F)c(Br)c1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 7/20 0.53
EPAS1 Q99814 1/20 0.51
TRPA1 O75762 6/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.43
SLC22A12 Q96S37 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15067944 0.90 PTGDR2 (0.53) BRD4EPAS1TRPA1PTGDR2
SCHEMBL15067741 0.86 BRD4 (0.54) BRD4EPAS1TRPA1PTGDR2
SCHEMBL21190911 0.83 BRD4 (0.56) BRD4EPAS1TRPA1PTGDR2SLC22A12
SCHEMBL16650562 0.81 TRPA1 (0.49) EPAS1TRPA1
SCHEMBL16650802 0.79 EPAS1 (0.72) BRD4EPAS1
SCHEMBL15068104 0.79 BRD4 (0.54) BRD4EPAS1TRPA1
SCHEMBL21652768 0.79 EPAS1 (0.43) BRD4EPAS1TRPA1PTGDR2
SCHEMBL21191082 0.78 BRD4 (0.55) BRD4EPAS1TRPA1
SCHEMBL21190939 0.77 BRD4 (0.46) BRD4EPAS1TRPA1
SCHEMBL15067629 0.76 PKM (0.43) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230158039-A1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2023-05-25 US disclosed
US-20210236508-A1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2021-08-05 US disclosed
CN-106986872-B Bromodomain inhibitors 艾伯维公司 2020-04-21 CN disclosed
US-20180296566-A1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2018-10-18 US disclosed
EP-2797918-B1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2017-11-29 EP disclosed
US-20160143916-A1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2016-05-26 US disclosed
US-9296741-B2 Bromodomain inhibitors ABBVIE INC. (US) 2016-03-29 US disclosed
EP-2797918-A1 BROMODOMAIN INHIBITORS AbbVie Inc. (US) 2014-11-05 EP disclosed
US-20140162971-A1 BROMODOMAIN INHIBITORS ABBVIE INC. 2014-06-12 US disclosed
WO-2013097601-A1 BROMODOMAIN INHIBITORS ABBVIE INC. (US) 2013-07-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180296566-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885EPAS1 2025/4885TRPA1 3858/4885
US-20140162971-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885EPAS1 2025/4885TRPA1 3858/4885
US-20230158039-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885EPAS1 2025/4885TRPA1 3858/4885
US-20160143916-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885EPAS1 2025/4885TRPA1 3858/4885
US-20210236508-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885EPAS1 2025/4885TRPA1 3858/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.