SCHEMBL15074479

SCHEMBL15074479

CC(C)[S+]([O-])c1cncc(Br)c1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
PTK2 Q05397 1/20 0.33
CYP2A6 P11509 2/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
KDM4E B2RXH2 2/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1403825 0.78 POLB (0.36) POLBHCAR2PTK2CYP2A6HTT
SCHEMBL19674652 0.73 POLB (0.33) POLBHCAR2PTK2CYP2A6HTT
SCHEMBL30639795 0.73 POLB (0.37) POLBHCAR2PTK2HTTRAB9A
SCHEMBL23943395 0.72 ALDH1A1 (0.41) RAB9AALDH1A1MAPTMAPK1
SCHEMBL19674732 0.69 KDM4E (0.38) POLBHCAR2HTTRAB9AKDM4E
SCHEMBL16099522 0.69 CYP2A6 (0.38) CYP2A6ALDH1A1MAPK1
SCHEMBL19674604 0.68 POLB (0.30) POLBHCAR2
SCHEMBL23087851 0.68 HTT (0.42) POLBHCAR2PTK2CYP2A6HTT
SCHEMBL14516919 0.67
SCHEMBL19082518 0.67 ALDH1A1 (0.38) CYP2A6HTTKDM4ELMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3371170-B1 INDOLIN-2-ONE DERIVATIVES USEFUL IN THE TREATMENT OF CNS DISEASES HOFFMANN LA ROCHE (CH) 2019-07-31 EP disclosed
WO-2013093849-A1 DIHYDRO-BENZO-OXAZINE AND DIHYDRO-PYRIDO-OXAZINE DERIVATIVES NOVARTIS AG (CH) 2013-06-27 WO disclosed