SCHEMBL15074751

SCHEMBL15074751

COc1cc(OC)cc(-n2c3ccc(-n4c5ccccc5c5ccccc54)cc3c3cc(-n4c5ccccc5c5ccccc54)ccc32)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.54
KDM4E B2RXH2 4/20 0.54
L3MBTL1 Q9Y468 4/20 0.54
ALDH1A1 P00352 4/20 0.54
HPGD P15428 3/20 0.54
HTT P42858 2/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
HSD17B10 Q99714 1/20 0.54
ATM Q13315 2/20 0.46
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
HCRTR1 O43613 1/20 0.42
RAB9A P51151 1/20 0.42
PAX8 Q06710 1/20 0.42
HTR6 P50406 1/20 0.41
RXFP1 Q9HBX9 2/20 0.40
EDNRA P25101 1/20 0.39
TP53 P04637 1/20 0.38
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734122 0.91 L3MBTL1 (0.54) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL29386 0.90 MAPT (0.58) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL8739926 0.89 KDM4E (0.57) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL22894292 0.89 KDM4E (0.57) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL14407598 0.85 MAPT (0.70) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL17691641 0.84 KDM4E (0.53) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL23264343 0.84 KDM4E (0.58) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL28988538 0.83 MAPT (0.68) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL30352484 0.83 MAPT (0.68) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL16171511 0.82 MAPT (0.50) MAPTKDM4EL3MBTL1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190259964-A1 ORGANIC SEMICONDUCTOR COMPOSITION AND SEMICONDUCTING LAYER OBTAINED THEREFROM SOLVAY SA (BE) 2019-08-22 US disclosed
WO-2017216168-A1 ORGANIC SEMICONDUCTOR COMPOSITION AND SEMICONDUCTING LAYER OBTAINED THEREFROM SOLVAY SA (BE) 2017-12-21 WO disclosed
EP-3257849-A1 ORGANIC SEMICONDUCTOR COMPOSITION AND SEMICONDUCTING LAYER OBTAINED THEREFROM Solvay SA (BE) 2017-12-20 EP disclosed
WO-2013096832-A2 SMALL MOLECULE CROSSLINKABLE TRISCARBAZOLE HOLE TRANSPORT MATERIALS GEORGIA TECH RESEARCH CORPORATION (US) 2013-06-27 WO disclosed
WO-2013096921-A1 NON-CROSSLINKED POLYSTYRENE TRISCARBAZOLE HOLE TRANSPORT MATERIALS GEORGIA TECH RESEARCH CORPORATION (US) 2013-06-27 WO disclosed