SCHEMBL15080293

SCHEMBL15080293

CNC1=NC2(CCc3cc(-c4c(C)nn(C)c4C)ccc3C2)CO1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.35
BRD4 O60885 2/20 0.34
HTR1A P08908 1/20 0.34
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
PIK3CD O00329 1/20 0.32
PIK3CG P48736 1/20 0.32
MAP4K1 Q92918 1/20 0.32
CREBBP Q92793 1/20 0.32
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12203461 0.88 BRD4 (0.36) HTR7BRD4HTR1APRMT5WDR77
SCHEMBL7916585 0.86 TAAR1 (0.42) HTR7BRD4HTR1APRMT5WDR77
SCHEMBL15080294 0.81 OTUD7B (0.38) BRD4PIK3CDPIK3CG
SCHEMBL15080312 0.78 CYP3A4 (0.36) BACE1
SCHEMBL7928716 0.77 BRD4 (0.37) HTR7BRD4HTR1APRMT5WDR77
SCHEMBL15080311 0.77 BACE1 (0.40) BACE1
SCHEMBL7922955 0.76 PRMT5 (0.36) HTR7BRD4HTR1APRMT5WDR77
SCHEMBL7930498 0.71 PIK3CD (0.40) HTR7BRD4HTR1APRMT5WDR77
SCHEMBL12203463 0.68 OTUD7B (0.40) BRD4PIK3CDPIK3CG
SCHEMBL7924981 0.67 BRD4 (0.47) BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8476274-B2 Biaryl spiroaminooxazoline analogues as Alpha2C adrenergic receptor modulators MERCK SHARP & DOHME CORP. (US) 2013-07-02 US disclosed