SCHEMBL15080504

SCHEMBL15080504

CCCCc1csc(N(C)C)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
ADRB2 P07550 2/20 0.43
ADRB1 P08588 2/20 0.43
ADRB3 P13945 2/20 0.43
KCNH2 Q12809 1/20 0.36
NOS2 P35228 1/20 0.36
SLC6A3 Q01959 1/20 0.34
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
LMNA P02545 2/20 0.32
ABCB11 O95342 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
SCN1A P35498 1/20 0.32
SCN2A Q99250 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
SCN3A Q9NY46 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13947093 0.89 MEN1 (0.53) MEN1KMT2AADRB2ADRB1ADRB3
SCHEMBL12800176 0.84 ADRB2 (0.39) MEN1KMT2AADRB2ADRB1ADRB3
SCHEMBL13662109 0.80 MEN1 (0.56) MEN1KMT2AADRB2ADRB1ADRB3
SCHEMBL9386347 0.79 MEN1 (0.47) MEN1KMT2AADRB2ADRB1ADRB3
SCHEMBL11991390 0.76 MEN1 (0.49) MEN1KMT2AADRB2ADRB1ADRB3
SCHEMBL723608 0.75 ADRB2 (0.41) MEN1KMT2AADRB2ADRB1ADRB3
SCHEMBL7176303 0.75 MEN1 (0.54) MEN1KMT2AMAPTRAB9ALMNA
SCHEMBL7179302 0.75 KMT2A (0.50) MEN1KMT2AMAPTRAB9ALMNA
SCHEMBL18381553 0.75 MEN1 (0.50) MEN1KMT2AMAPTRAB9ALMNA
SCHEMBL2631523 0.75 PKM (0.45) MEN1KMT2AKCNH2NOS2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8912182-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-12-16 US disclosed
US-8541402-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-09-24 US disclosed
US-8476257-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-07-02 US disclosed