SCHEMBL1508089

SCHEMBL1508089

CCCOc1ccc2c(Cl)nc(C(=O)NCC(=O)O)c(O)c2c1I

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 17/20 0.51
BBOX1 O75936 2/20 0.51
FTO Q9C0B1 2/20 0.51
THRA P10827 5/20 0.48
THRB P10828 5/20 0.48
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
ASPH Q12797 1/20 0.40
KDM8 Q8N371 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1841936 0.85 EGLN1 (0.56) EGLN1BBOX1FTOTHRATHRB
SCHEMBL5318572 0.84 EGLN1 (0.50) EGLN1BBOX1FTOTHRATHRB
SCHEMBL4409796 0.82 EGLN1 (0.64) EGLN1BBOX1FTOTHRATHRB
SCHEMBL4411746 0.81 EGLN1 (0.61) EGLN1BBOX1FTOTHRATHRB
SCHEMBL522269 0.78 THRA (0.70) EGLN1BBOX1FTOTHRATHRB
SCHEMBL522867 0.78 THRA (0.64) EGLN1BBOX1FTOTHRATHRB
SCHEMBL4973457 0.77 EGLN1 (0.58) EGLN1BBOX1FTOTHRATHRB
SCHEMBL5325511 0.77 EGLN1 (0.61) EGLN1BBOX1FTOTHRATHRB
SCHEMBL5027666 0.74 EGLN1 (0.68) EGLN1BBOX1FTOTHRATHRB
SCHEMBL4411721 0.74 EGLN1 (0.58) EGLN1BBOX1FTOTHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295060-A2 Stabilization of hypoxia inducible factor (HIF) alpha FIBROGEN, INC. (US) 2011-03-16 EP disclosed