SCHEMBL15083063

SCHEMBL15083063

O=C(O)c1cc(-c2ccncn2)ns1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.41
CAMKK2 Q96RR4 1/20 0.40
SCD O00767 2/20 0.36
SCD5 Q86SK9 2/20 0.36
KMO O15229 2/20 0.35
GRM1 Q13255 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CDC7 O00311 1/20 0.34
P2RX7 Q99572 1/20 0.33
NAPRT Q6XQN6 1/20 0.33
JAK2 O60674 1/20 0.33
GSK3B P49841 1/20 0.33
LATS1 O95835 1/20 0.33
LATS2 Q9NRM7 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27905752 0.89 CYP3A4 (0.39) CYP3A4CAMKK2SCDSCD5GRM1
SCHEMBL12571315 0.79 KDM4E (0.57) CYP3A4KDM4ENAPRT
SCHEMBL31561147 0.79 KDM4E (0.57) CYP3A4KDM4ENAPRT
SCHEMBL15083062 0.78 MAPK14 (0.43) GRM1KDM4ECDC7NAPRT
SCHEMBL12571319 0.75 KDM4E (0.43) CYP3A4SCD5KDM4ECDC7NAPRT
SCHEMBL11889639 0.73 KDM4E (0.63) KDM4E
SCHEMBL12571320 0.73 KDM4E (0.41) CYP3A4KDM4ENAPRT
SCHEMBL27905755 0.72 GSK3B (0.41) CYP3A4CDC7GSK3BLATS1LATS2
SCHEMBL12571404 0.71 ALDH1A1 (0.48) CAMKK2SCDSCD5KMOKDM4E
SCHEMBL12571313 0.71 DHODH (0.45) KDM4EP2RX7NAPRT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8884020-B2 Indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2014-11-11 US disclosed
EP-2610244-A1 Indole compounds Ironwood Pharmaceuticals, Inc. (US) 2013-07-03 EP disclosed