SCHEMBL15083062

SCHEMBL15083062

O=C(O)c1cc(-c2ccncc2)ns1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.43
DHODH Q02127 1/20 0.41
NAPRT Q6XQN6 1/20 0.41
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
CDC7 O00311 3/20 0.38
DBF4 Q9UBU7 3/20 0.38
CASP1 P29466 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
CYP46A1 Q9Y6A2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768523 0.87 CASP1 (0.38) MAPK14DHODHALDH1A1GAACDC7
SCHEMBL6843818 0.85 TP53 (0.44) DHODHALDH1A1GAAMAPTKDM4E
SCHEMBL15083064 0.83 HCAR2 (0.43) MAPK14HDAC4MKNK1MKNK2
SCHEMBL2722584 0.81 MKNK1 (0.58) DHODHALDH1A1GAAHDAC3HDAC4
SCHEMBL28093059 0.81 CA12 (0.49) MAPK14DHODHALDH1A1MAPTKDM4E
SCHEMBL6740513 0.81 ALAD (0.51) ALDH1A1CASP1MAPTKDM4EKMT2A
SCHEMBL6668534 0.81 ALAD (0.51)
SCHEMBL4553247 0.80 PPARD (0.44) CASP1MAPT
SCHEMBL15083063 0.78 CYP3A4 (0.41) NAPRTCDC7GRM1KDM4E
SCHEMBL11000258 0.77 ALPL (0.52) ALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8884020-B2 Indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2014-11-11 US disclosed
EP-2610244-A1 Indole compounds Ironwood Pharmaceuticals, Inc. (US) 2013-07-03 EP disclosed