SCHEMBL15085525

SCHEMBL15085525

COc1ccc(Cn2ccn(C)c2=[Pt])cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.49
TP53 P04637 2/20 0.49
LMNA P02545 1/20 0.49
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
ALOX15 P16050 1/20 0.46
CMA1 P23946 1/20 0.46
LPO P22079 2/20 0.46
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
SIGMAR1 Q99720 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
POLB P06746 1/20 0.40
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2194410 0.85 MAPT (0.39) MAPTTP53LMNAKDM4EALDH1A1
SCHEMBL2195709 0.85 MAPT (0.41) MAPTTP53LMNAKDM4EALDH1A1
SCHEMBL2198394 0.84 MAPT (0.42) MAPTTP53LMNAKDM4EALDH1A1
SCHEMBL2194976 0.84 SIGMAR1 (0.44) MAPTTP53LMNALPOCYP11B1
SCHEMBL2195090 0.84 MAPT (0.41) MAPTTP53LMNAALDH1A1LPO
SCHEMBL2193843 0.83 MET (0.43) MAPTTP53LMNAKDM4EALDH1A1
SCHEMBL2195198 0.83 SIGMAR1 (0.40) MAPTTP53LMNAALDH1A1SIGMAR1
SCHEMBL2196792 0.83 MAPT (0.40) MAPTTP53LMNAALDH1A1SIGMAR1
SCHEMBL2195985 0.83 MAPT (0.38) MAPTTP53LMNAKDM4EALDH1A1
SCHEMBL2194293 0.83 MAPT (0.39) MAPTTP53LMNAALDH1A1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8980875-B2 Platinum-N-heterocyclic carbene derivatives, preparation thereof and therapeutic use thereof CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2015-03-17 US claimed
US-20130338128-A1 PLATINUM-N-HETEROCYCLIC CARBENE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2013-12-19 US claimed
US-8481522-B2 Platinum-N-heterocyclic carbene derivatives, preparation thereof and therapeutic use thereof SANOFI (FR) 2013-07-09 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130338128-A1 PLATINUM-N-HETEROCYCLIC CARBENE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SCO2, C3AR1, IDH1 MAPT 4712/4885TP53 1327/4885LMNA 2301/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.