SCHEMBL1508765

SCHEMBL1508765

C[C@H]1CN(C(=O)C(F)(F)F)C2(CC2)CN1C(=O)[C@@H]1C[C@](C)(O[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)CN1C(=O)OC(C)(C)C

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RORC P51449 10/20 0.31
HDAC1 Q13547 1/20 0.30
GPR119 Q8TDV5 3/20 0.30
TACR1 P25103 2/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1508993 0.83
SCHEMBL1508995 0.83
SCHEMBL14802189 0.79
SCHEMBL2490403 0.79
SCHEMBL1508660 0.78 RORC (0.37) RORCGPR119
SCHEMBL1508767 0.77
SCHEMBL1509094 0.74 HSD17B10 (0.46)
SCHEMBL2527201 0.74
SCHEMBL1509084 0.74 HSD17B10 (0.46)
SCHEMBL1509097 0.74 CYP1A2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298778-A1 IMIDAZOTHIAZOLE DERIVATIVE HAVING 4,7-DIAZASPIROÝ2.5¨OCTANE RING STRUCTURE Daiichi Sankyo Company, Limited (JP) 2011-03-23 EP disclosed