SCHEMBL15087906

SCHEMBL15087906

COCc1cc(-c2ccnc(Cl)n2)cs1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2E1 P05181 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2A6 P11509 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP4B1 P13584 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP3A5 P20815 1/20 0.34
CYP2A7 P20853 1/20 0.34
CYP3A7 P24462 1/20 0.34
CYP2F1 P24903 1/20 0.34
CYP2C18 P33260 1/20 0.34
CYP2C19 P33261 1/20 0.34
CYP2J2 P51589 1/20 0.34
CYP4F2 P78329 1/20 0.34
CYP4F8 P98187 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1108279 0.84 ALDH1A1 (0.37) AAK1KMOSREBF2MAPTKDM4E
SCHEMBL1097848 0.81 AAK1 (0.34) AAK1KMONPC1SREBF2MAPT
SCHEMBL1097565 0.81 GAA (0.31)
SCHEMBL15087871 0.75 DPP4 (0.44) CYP1A2CYP2E1CYP2D6CYP2A6CYP2C9
SCHEMBL15087883 0.75 DAO (0.37) AAK1CYP1A1CYP1A2CYP2E1CYP3A4
SCHEMBL15577810 0.75 DYRK1A (0.46) DYRK1ACLK4DYRK1BCLK1CLK2
SCHEMBL15087879 0.73 DYRK1A (0.44) DYRK1ACLK4DYRK1BCLK1KMO
SCHEMBL1098764 0.71 CYP2A6 (0.34) AAK1CYP2A6KMOMEN1KMT2A
SCHEMBL24638508 0.70 IKBKE (0.38) AAK1KMONPC1MAPTMEN1
SCHEMBL27111217 0.70 MAPT (0.47) CYP1A1CYP1A2CYP2E1CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130172338-A1 OXYGEN LINKED PYRIMIDINE DERIVATIVES CELL THERAPEUTICS, INC. (US) 2013-07-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130172338-A1 OXYGEN LINKED PYRIMIDINE DERIVATIVES DPYD, TK2, TK1 AAK1 996/4885CYP1A1 2156/4885CYP1A2 2142/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.