SCHEMBL15090591

SCHEMBL15090591

O=C(c1ccc(C(=O)NC2C3CC4CC2CC(O)(C4)C3)c(OC2CCOCC2)c1)c1ccccc1F

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 19/20 0.47
HSD11B2 P80365 1/20 0.46
KAT2B Q92831 1/20 0.44
BAZ2B Q9UIF8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15100752 1.00 HSD11B1 (0.47) HSD11B1HSD11B2KAT2BBAZ2B
SCHEMBL257359 0.93 HSD11B1 (0.48) HSD11B1HSD11B2
SCHEMBL15090633 0.93 HSD11B1 (0.48) HSD11B1HSD11B2
SCHEMBL15090539 0.92 HSD11B1 (0.47) HSD11B1HSD11B2
SCHEMBL10046962 0.92 HSD11B1 (0.47) HSD11B1HSD11B2
SCHEMBL15198837 0.92 HSD11B1 (0.47) HSD11B1HSD11B2
SCHEMBL10046793 0.87 HSD11B1 (0.51) HSD11B1HSD11B2
SCHEMBL257370 0.86 KAT2B (0.41) HSD11B1HSD11B2KAT2BBAZ2B
SCHEMBL15090525 0.83 HSD11B1 (0.49) HSD11B1HSD11B2
SCHEMBL256767 0.83 HSD11B1 (0.49) HSD11B1HSD11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895552-B2 Cyclic amide derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2014-11-25 US disclosed
US-20130217692-A1 CYCLIC AMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2013-08-22 US disclosed
EP-2612848-A1 CYCLIC AMIDE DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2013-07-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130217692-A1 CYCLIC AMIDE DERIVATIVE HDAC10, H1-10, H1-0 HSD11B1 583/4885HSD11B2 915/4885KAT2B 140/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.