SCHEMBL15201250

SCHEMBL15201250

Cc1ccc(N)cc1Nc1nccc(=O)[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.45
BCR P11274 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LCK P06239 1/20 0.41
DOT1L Q8TEK3 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
MAPKAPK2 P49137 1/20 0.35
RPS6KA3 P51812 1/20 0.35
CSNK2A1 P68400 1/20 0.35
PLK3 Q9H4B4 1/20 0.35
LMNA P02545 1/20 0.34
ALDH1A1 P00352 1/20 0.34
AURKA O14965 1/20 0.34
AURKB Q96GD4 1/20 0.34
ADRA2A P08913 1/20 0.33
ADRA2C P18825 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15201247 0.80 KMT2A (0.68) MEN1KMT2ASMN1; SMN2TAAR1ALDH1A1
SCHEMBL15201324 0.78 TSHR (0.48) KMT2ASMN1; SMN2ALDH1A1
SCHEMBL15201246 0.74 KMT2A (0.43) ABL1BCRMEN1KMT2ALCK
SCHEMBL6295526 0.74 MAPT (0.51) MEN1KMT2ADOT1LPDE3BPDE3A
SCHEMBL5815619 0.73 ABL1 (0.45) ABL1BCR
SCHEMBL15201330 0.73 ABL1 (0.55) ABL1BCRKMT2AALDH1A1AURKA
SCHEMBL15201248 0.71 ABL1 (0.40) ABL1BCRMEN1KMT2ALCK
SCHEMBL2616948 0.70 ABL1 (0.59) ABL1BCRMEN1KMT2ALCK
SCHEMBL13316450 0.70 KARS1 (0.50) ABL1BCRMEN1KMT2ALCK
Hydrochloric Acid SCHEMBL5548680 0.69 ABL1 (0.58) ABL1BCRMEN1KMT2ALCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013120852-A1 INTERMEDIATES FOR A NOVEL PROCESS OF PREPARING IMATINIB AND RELATED TYROSINE KINASE INHIBITORS GRINDEKS, A JOINT STOCK COMPANY (LV) 2013-08-22 WO claimed
WO-2013120852-A1 INTERMEDIATES FOR A NOVEL PROCESS OF PREPARING IMATINIB AND RELATED TYROSINE KINASE INHIBITORS GRINDEKS, A JOINT STOCK COMPANY (LV) 2013-08-22 WO disclosed
WO-2013120852-A1 INTERMEDIATES FOR A NOVEL PROCESS OF PREPARING IMATINIB AND RELATED TYROSINE KINASE INHIBITORS GRINDEKS, A JOINT STOCK COMPANY (LV) 2013-08-22 WO disclosed