SCHEMBL15211432

SCHEMBL15211432

CC(=O)c1c(O)ccc2c(CCl)cc(=O)oc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 6/20 0.68
ALDH1A1 P00352 4/20 0.59
HPGD P15428 3/20 0.59
LMNA P02545 2/20 0.59
PON1 P27169 1/20 0.56
CA9 Q16790 1/20 0.52
MAOB P27338 3/20 0.49
KDM4E B2RXH2 5/20 0.48
GLA P06280 2/20 0.48
PTPN1 P18031 1/20 0.43
GAA P10253 2/20 0.43
ATM Q13315 1/20 0.43
ERAP1 Q9NZ08 1/20 0.43
MEN1 O00255 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MGAM O43451 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL876286 0.81 MCL1 (0.73) MCL1ALDH1A1HPGDPON1CA9
SCHEMBL28065506 0.81 MCL1 (1.00) MCL1ALDH1A1HPGDLMNAPON1
SCHEMBL15211418 0.80 MCL1 (0.75) MCL1ALDH1A1HPGDPON1MAOB
SCHEMBL29749855 0.80 MAOB (0.67) MCL1ALDH1A1HPGDLMNACA9
SCHEMBL4383562 0.80 MAOB (0.67) MCL1ALDH1A1HPGDLMNACA9
SCHEMBL31454846 0.78 ERAP1 (0.54) MCL1ALDH1A1HPGDLMNACA9
SCHEMBL15211319 0.77 MCL1 (0.66) MCL1ALDH1A1HPGDPON1MAOB
SCHEMBL31454860 0.75 ALDH1A1 (0.58) MCL1ALDH1A1HPGDLMNAMAOB
SCHEMBL31454864 0.74 MCL1 (0.49) MCL1ALDH1A1HPGDLMNAMAOB
SCHEMBL31454884 0.73 ALDH1A1 (0.65) MCL1ALDH1A1HPGDLMNAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2838891-B1 AROMATIC RING COMPOUND AS GHRELIN O-ACYLTRANSFERASE INHIBITOR TAKEDA PHARMACEUTICALS CO (JP) 2017-08-02 EP disclosed
US-9238639-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-01-19 US disclosed
EP-2838891-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-02-25 EP disclosed
CN-104254525-A Aromatic ring compound TAKEDA PHARMACEUTICAL 2014-12-31 CN disclosed
WO-2013125732-A1 AROMATIC RING COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-29 WO disclosed