SCHEMBL15212266

SCHEMBL15212266

CCOC(=O)c1cnc(SC)nc1C.CSc1ncc(C(=O)O)c(C)n1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.60
TDP1 Q9NUW8 2/20 0.60
POLB P06746 1/20 0.60
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
SYK P43405 2/20 0.54
MAPT P10636 5/20 0.53
HPGD P15428 2/20 0.53
KDM4E B2RXH2 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
NFKB1 P19838 2/20 0.51
NFKB2 Q00653 2/20 0.51
RELA Q04206 2/20 0.51
LMNA P02545 1/20 0.51
FOS P01100 1/20 0.51
JUN P05412 1/20 0.51
HTT P42858 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
RAB9A P51151 2/20 0.50
MAPK1 P28482 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29897636 0.94 MEN1 (0.64) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL423187 0.94 MEN1 (0.64) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL4762536 0.87 HTT (0.55) POLBMEN1KMT2AHPGDKDM4E
SCHEMBL24340549 0.84 MAPT (0.55) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL20649220 0.84 MEN1 (0.63) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL3278294 0.83 MEN1 (0.61) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL31148410 0.83 MEN1 (0.61) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL31148360 0.82 ALDH1A1 (0.60) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL13696640 0.82 ALDH1A1 (0.60) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL2908655 0.81 RAB9A (0.56) ALDH1A1POLBMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817308-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES AbbVie Inc. (US) 2014-12-31 EP disclosed
WO-2013126656-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES ABBVIE INC. (US) 2013-08-29 WO disclosed