SCHEMBL15212500

SCHEMBL15212500

C=Cc1c[nH]c(=O)c2cncnc12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DPYD Q12882 1/20 0.40
AURKA O14965 1/20 0.32
TTK P33981 1/20 0.32
AURKB Q96GD4 1/20 0.32
INCENP Q9NQS7 1/20 0.32
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.31
ADORA2A P29274 1/20 0.31
SLC6A4 P31645 1/20 0.31
ADRA1A P35348 1/20 0.31
XDH P47989 1/20 0.31
RAB9A P51151 1/20 0.31
BLM P54132 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CHEK1 O14757 1/20 0.30
RPS6KA5 O75582 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16652137 0.75 GSK3B (0.37) AURKATTKAURKBINCENPLMNA
SCHEMBL29722432 0.75 MAPK1 (0.35) DPYDAURKATTKAURKBINCENP
SCHEMBL18980749 0.75 MAPK1 (0.35) DPYDAURKATTKAURKBINCENP
SCHEMBL30208802 0.73 RPS6KA5 (0.42) DPYDCHEK1RPS6KA5
SCHEMBL30970570 0.71 AURKA (0.32) AURKATTKAURKBINCENP
SCHEMBL4212717 0.68 PARP1 (0.50) DPYDAURKBLMNARAB9ABLM
SCHEMBL13725532 0.62 CCNT1 (0.40)
SCHEMBL3434268 0.62 KMT2A (0.54) CHEK1RPS6KA5
SCHEMBL29955602 0.62 KMT2A (0.54) CHEK1RPS6KA5
SCHEMBL30812401 0.61 AURKA (0.34) AURKATTKAURKBINCENP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817308-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES AbbVie Inc. (US) 2014-12-31 EP claimed
WO-2013126656-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES ABBVIE INC. (US) 2013-08-29 WO claimed
EP-2817308-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES AbbVie Inc. (US) 2014-12-31 EP disclosed
WO-2013126656-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES ABBVIE INC. (US) 2013-08-29 WO disclosed