SCHEMBL15212935

SCHEMBL15212935

O=C(O)N1CCN(Cc2cc(Br)c3c([AsH2])ncnn23)CC1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACVRL1 P37023 9/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
FAAH O00519 7/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14888176 0.87 ACVRL1 (0.46) ACVRL1KDM4EALDH1A1LMNA
SCHEMBL5137764 0.74 ACVRL1 (0.46) ACVRL1
SCHEMBL57703 0.72 FGFR1 (0.48) ACVRL1
SCHEMBL5077251 0.70 ACVRL1 (0.38) ACVRL1KDM4EALDH1A1
SCHEMBL15019846 0.68 FGFR1 (0.42) ACVRL1
SCHEMBL15020405 0.68 FGFR1 (0.38) ACVRL1LMNA
SCHEMBL16011267 0.68 ACVRL1 (0.62) ACVRL1KDM4EALDH1A1
SCHEMBL59608 0.67 ACVRL1 (0.64) ACVRL1KDM4E
SCHEMBL15019887 0.65 FGFR1 (0.39) ACVRL1
SCHEMBL15019263 0.65 FGFR1 (0.36) ACVRL1ALDH1A1LMNAFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817311-A1 SUBSTITUTED BENZOTHIENYL-PYRROLOTRIAZINES AND USES THEREOF Bayer Intellectual Property GmbH (DE) 2014-12-31 EP disclosed
WO-2013124316-A1 SUBSTITUTED BENZOTHIENYL-PYRROLOTRIAZINES AND USES THEREOF BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-08-29 WO disclosed