SCHEMBL15214952

SCHEMBL15214952

CC(C)S(=O)(=O)c1ccccc1Nc1nc(N)nc2ccnn12

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 15/20 0.41
CDK7 P50613 14/20 0.41
ADRA2A P08913 1/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
ALK Q9UM73 2/20 0.37
TTK P33981 1/20 0.36
HDAC1 Q13547 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1070192 0.85 CDK7 (0.38) CDK9CDK7ADRA2AADRA1DADRA1A
SCHEMBL1070526 0.84 CDK7 (0.38) CDK9CDK7ADRA2AADRA1DADRA1A
SCHEMBL1072883 0.79 KCNN3 (0.54) CDK9CDK7ALK
SCHEMBL12364043 0.75 PTK2 (0.42) ALKHDAC1
SCHEMBL12364041 0.74 ALK (0.59) CDK9CDK7ALK
SCHEMBL11916291 0.73 ALK (0.61) ALKTTK
SCHEMBL12364046 0.73 ALK (0.48) ALK
SCHEMBL3949151 0.72 CDK7 (0.51) CDK9CDK7ALKHDAC1
SCHEMBL12364037 0.72 ALK (0.57) ALK
SCHEMBL12364040 0.71 KMT2A (0.41) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8518931-B2 Compounds and compositions as kinase inhibitors IRM LLC (BM) 2013-08-27 US disclosed