SCHEMBL1521573

SCHEMBL1521573

c1cnc(Cc2cnccn2)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.43
CYP3A4 P08684 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HRH1 P35367 9/20 0.37
CYP2D6 P10635 8/20 0.37
KCNH2 Q12809 3/20 0.37
CHRM1 P11229 1/20 0.37
HTR2A P28223 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NAPRT Q6XQN6 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
VNN1 O95497 1/20 0.36
BAZ2B Q9UIF8 1/20 0.36
ADORA3 P0DMS8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL980114 0.85
SCHEMBL16598063 0.84 HRH3 (0.53) CYP3A4CYP1A2CYP2C9CYP2C19HRH1
SCHEMBL16598474 0.82 KCNH3 (0.36) HSP90AA1CYP3A4HDAC3HDAC1HDAC2
SCHEMBL16597995 0.82 CYP2D6 (0.38) HSP90AA1CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL13171962 0.81 CYP11B1 (0.37) HSP90AA1CYP3A4HDAC3HDAC1HDAC2
SCHEMBL14274076 0.81 HRH1 (0.36) HSP90AA1CYP3A4HDAC3HDAC1HDAC2
SCHEMBL18674013 0.79 HRH1 (0.41) CYP3A4HDAC6CYP1A2CYP2C9CYP2C19
SCHEMBL3048473 0.79 ALDH1A1 (0.50) CYP3A4CYP1A2CYP2C9CYP2C19HRH1
SCHEMBL12431 0.78
SCHEMBL284256 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012112758-A2 VIRTUAL HYDROGEN STORAGE PROCESSES AND RELATED CATALYSTS AND SYSTEMS YALE UNIVERSITY (US) 2012-08-23 WO claimed
US-7901491-B2 Hydrogen storage material and related system GENERAL ELECTRIC COMPANY (US) 2011-03-08 US claimed
US-20090246575-A1 HYDROGEN STORAGE MATERIAL AND RELATED SYSTEM GENERAL ELECTRIC COMPANY (US) 2009-10-01 US claimed
US-20080248339-A1 METHOD AND APPARATUS FOR ELECTROCHEMICAL ENERGY CONVERSION GENERAL ELECTRIC COMPANY (US) 2008-10-09 US claimed
US-20080248345-A1 METHOD AND APPARATUS FOR ELECTROCHEMICAL ENERGY CONVERSION GENERAL ELECTRIC COMPANY (US) 2008-10-09 US claimed
WO-2013103724-A1 2- (TERT - BUTOXY) -2- (7 -METHYLQUINOLIN- 6 - YL) ACETIC ACID DERIVATIVES FOR TREATING AIDS GILEAD SCIENCES, INC. (US) 2013-07-11 WO disclosed
WO-2012112758-A2 VIRTUAL HYDROGEN STORAGE PROCESSES AND RELATED CATALYSTS AND SYSTEMS YALE UNIVERSITY (US) 2012-08-23 WO disclosed
US-7901491-B2 Hydrogen storage material and related system GENERAL ELECTRIC COMPANY (US) 2011-03-08 US disclosed
US-20100038592-A1 COMPOSITION AND LIGHT-EMITTING ELEMENT COMPRISING THE COMPOSITION SUMATION CO., LTD. (JP) 2010-02-18 US disclosed
US-20100038592-A1 COMPOSITION AND LIGHT-EMITTING ELEMENT COMPRISING THE COMPOSITION SUMATION CO., LTD. (JP) 2010-02-18 US disclosed
US-20090246575-A1 HYDROGEN STORAGE MATERIAL AND RELATED SYSTEM GENERAL ELECTRIC COMPANY (US) 2009-10-01 US disclosed
US-20080248339-A1 METHOD AND APPARATUS FOR ELECTROCHEMICAL ENERGY CONVERSION GENERAL ELECTRIC COMPANY (US) 2008-10-09 US disclosed
US-20080248345-A1 METHOD AND APPARATUS FOR ELECTROCHEMICAL ENERGY CONVERSION GENERAL ELECTRIC COMPANY (US) 2008-10-09 US disclosed
EP-1830858-A2 3, 6-BICYCLOLIDES Enanta Pharmaceuticals, Inc. (US) 2007-09-12 EP disclosed
WO-2006063039-A2 3, 6-BICYCLOLIDES ENANTA PHARMACEUTICALS, INC. (US) 2006-06-15 WO disclosed