SCHEMBL15216009

SCHEMBL15216009

COc1cc2ccn3cncc3c2cc1OC(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.44
QPCT Q16769 1/20 0.36
QPCTL Q9NXS2 1/20 0.36
MAPT P10636 3/20 0.36
PSMB1 P20618 2/20 0.34
PSMB5 P28074 2/20 0.34
MAOA P21397 2/20 0.34
PSMB2 P49721 1/20 0.34
PDE10A Q9Y233 3/20 0.33
PDE4A P27815 1/20 0.33
PDE4D Q08499 1/20 0.33
CYP17A1 P05093 1/20 0.33
TNF P01375 1/20 0.33
SUV39H2 Q9H5I1 2/20 0.33
SOS1 Q07889 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2777878 0.69 RPS6KB2 (0.44) IDO1MAPTPDE4APDE4DALDH1A1
SCHEMBL15216010 0.67 PSMB1 (0.34) PSMB1PSMB5PSMB2PDE10ATNF
SCHEMBL10651277 0.66 TNF (0.41) PSMB1PSMB5PSMB2PDE4APDE4D
SCHEMBL13409741 0.66 TNF (0.49) MAPTPDE10APDE4APDE4DTNF
SCHEMBL29702221 0.66 LRRK2 (0.48) MAPTPSMB1PSMB5PDE10APDE4A
SCHEMBL31207123 0.65 ALDH1A1 (0.43) MAPTMAOAPDE10APDE4APDE4D
SCHEMBL8315056 0.65 TLR8 (0.45) IDO1MAPTPDE10ASOS1ALDH1A1
SCHEMBL7413595 0.63 MAPT (0.40) MAPTMAOAPDE10APDE4APDE4D
SCHEMBL11535971 0.63 IDO1 (1.00) IDO1QPCTQPCTLMAPTALDH1A1
SCHEMBL25020508 0.62 IRAK4 (0.42) PSMB1PSMB5PSMB2PDE10APDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2435433-B1 (DIHYDRO)IMIDAZOISO[5,1-A]QUINOLINES AS FSH RECEPTOR AGONISTS FOR THE TREATMENT OF FERTILITY DISORDERS MERCK SHARP & DOHME (NL) 2013-08-28 EP disclosed