SCHEMBL1521650

SCHEMBL1521650

CC(C)(C)c1cc(NC(=O)Nc2cc(N3Cc4cnc(CN)cc4NC3=O)ccc2F)n(-c2ccccc2)n1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 14/20 0.51
MAPK13 O15264 11/20 0.51
MAPK12 P53778 11/20 0.51
MAPK11 Q15759 11/20 0.51
BRAF P15056 5/20 0.45
NTRK1 P04629 1/20 0.44
NTRK3 Q16288 1/20 0.44
NTRK2 Q16620 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1521548 0.91 MAPK14 (0.43) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1521555 0.79 MAPK14 (0.53) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1521814 0.79 MAPK14 (0.52) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1521965 0.78 MAPK14 (0.51) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1521946 0.77 ABL1 (0.52) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1521734 0.76 MAPK14 (0.51) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1011086 0.73 MAPK14 (0.70) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1521722 0.72 KCNJ6 (0.48) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1521661 0.70 KCNJ6 (0.47) MAPK14MAPK13MAPK12MAPK11BRAF
SCHEMBL1521906 0.70 KCNJ6 (0.46) MAPK14MAPK13MAPK12MAPK11BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7897762-B2 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2011-03-01 US claimed