SCHEMBL15232609

SCHEMBL15232609

O=C(O)/C=C/CNC(=O)c1cc(Br)c[nH]1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA6 P17658 3/20 0.57
KCNA3 P22001 3/20 0.57
KCNA4 P22459 3/20 0.57
KCNA5 P22460 2/20 0.57
PKM P14618 2/20 0.56
DAO P14920 2/20 0.52
CREBBP Q92793 1/20 0.51
VIP P01282 1/20 0.43
EGFR P00533 1/20 0.39
ERBB2 P04626 1/20 0.39
HRH3 Q9Y5N1 3/20 0.38
SCN9A Q15858 1/20 0.38
SCN3A Q9NY46 1/20 0.38
IDO1 P14902 2/20 0.37
ADRA2A P08913 1/20 0.37
ADRA1D P25100 1/20 0.37
KCNA2 P16389 1/20 0.36
NT5E P21589 1/20 0.36
MAP2K1 Q02750 1/20 0.36
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15228546 1.00 KCNA6 (0.57) KCNA6KCNA3KCNA4KCNA5PKM
SCHEMBL15243719 0.81 KCNA6 (0.51) KCNA6KCNA3KCNA4KCNA5PKM
SCHEMBL14843672 0.80 SMYD3 (0.49) KCNA6KCNA3KCNA4KCNA5KMT2A
SCHEMBL13036735 0.74 KCNA6 (0.67) KCNA6KCNA3KCNA4KCNA5PKM
SCHEMBL7845382 0.74 PKM (0.60) KCNA6KCNA3KCNA4KCNA5PKM
SCHEMBL21182348 0.73 KCNA6 (1.00) KCNA6KCNA3KCNA4KCNA5PKM
SCHEMBL23952430 0.72 CREBBP (0.67) KCNA6KCNA3KCNA4KCNA5PKM
SCHEMBL28746425 0.71 CREBBP (0.60) KCNA6KCNA3KCNA4KCNA5PKM
Keramadine SCHEMBL11123414 0.70 KCNA6 (0.64) KCNA6KCNA3KCNA4KCNA5PKM
Keramadine SCHEMBL11123417 0.70 KCNA6 (0.64) KCNA6KCNA3KCNA4KCNA5PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9394297-B2 Amides as pim inhibitors AMGEN INC. (US) 2016-07-19 US disclosed
US-20150329538-A1 AMIDES AS PIM INHIBITORS AMGEN INC. (US) 2015-11-19 US disclosed
WO-2014022752-A1 MACROCYCLES AS PIM INHIBITORS AMGEN INC. (US) 2014-02-06 WO disclosed
WO-2013130660-A1 AMIDES AS PIM INHIBITORS AMGEN INC. (US) 2013-09-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150329538-A1 AMIDES AS PIM INHIBITORS PIM1, PIM3, PIM2 KCNA6 2073/4885KCNA3 1736/4885KCNA4 2908/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.